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Found 20 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 2'
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)
Affinity DataIC50:  450nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50220547(4,5-Dibromo-1H-pyrrole-2-carboxylic acid [3-(2-ami...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456982(CHEMBL4208517)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50507839(PF-6305591 | Pf-06305591)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Kv1.2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456970(CHEMBL3261431)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456973(Clathrodin)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456971(CHEMBL4210636)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456977(CHEMBL3261430)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456976(CHEMBL4207745)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456975(CHEMBL4213446)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Rattus norvegicus)
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant rat Kv1.2(4) expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50067880(4-methoxy-7H-furo[3,2-g][1]benzopyran-7-one | 4-me...)
Affinity DataKd:  4.10E+4nMAssay Description:Blockade of peak K+ currents against Kv1.2 geneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50067878(9-Methoxy-furo[3',2':4,5]benzo[1,2-b][1,4]oxazin-3...)
Affinity DataKd:  5.90E+5nMAssay Description:Blockade of peak K+ currents against Kv1.2 geneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50182587(5-acetyl-4-(4'-chloro)benzyloxy-6-hydroxy-7-methox...)
Affinity DataEC50:  2.50E+3nMAssay Description:Effect on blockade of Kv1.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50182585(5-acetyl-7-(4'-bromo)benzyloxy-6-hydroxy-4-methoxy...)
Affinity DataEC50:  1.40E+3nMAssay Description:Effect on blockade of Kv1.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50182597(5-acetyl-4,7-benzyloxy-6-hydroxybenzofuran | CHEMB...)
Affinity DataEC50:  1.00E+4nMAssay Description:Effect on blockade of Kv1.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50067879(5-Methoxymethyl-3-methyl-furo[3,2-g]chromen-7-one ...)
Affinity DataKd:  1.80E+4nMAssay Description:Blockade of peak K+ currents against Kv1.2 geneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50067881(4,9-Diethoxy-furo[3,2-g]chromen-7-one | CHEMBL3429...)
Affinity DataKd:  2.30E+4nMAssay Description:Blockade of peak K+ currents against Kv1.2 geneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed